{"id":462,"date":"2019-12-02T10:38:17","date_gmt":"2019-12-02T02:38:17","guid":{"rendered":"http:\/\/www.broadbio.com\/?p=462"},"modified":"2019-12-02T10:38:17","modified_gmt":"2019-12-02T02:38:17","slug":"12021","status":"publish","type":"post","link":"http:\/\/www.broadbio.com\/archives\/462","title":{"rendered":"\u6cd5\u56fdalsachim\u7a33\u5b9a\u540c\u4f4d\u7d20\u6807\u8bb0\u7269"},"content":{"rendered":"<p>\u6cd5\u56fdAlsaChim\u662f\u63d0\u4f9b\u9ad8\u54c1\u8d28\u7a33\u5b9a\u540c\u4f4d\u7d20\u5185\u6807\u548c\u4e34\u5e8a\u8d28\u8c31\u68c0\u6d4b\u8bd5\u5242\u76d2\u4ea7\u54c1\uff0c\u5176\u4e2d\u5305\u542b13C, 15N, 2H\u7684\u7a33\u5b9a\u540c\u4f4d\u7d20\u6807\u8bb0\uff0c\u4ea7\u54c1\u00a013C, 15N\u6807\u8bb0\u7eaf\u5ea6&gt;99%\uff0c\u5176\u4e2d13C\u6807\u8bb0\u7684\u201c\u9ec4\u91d1\u6807\u51c6\u201d\u3002\u516c\u53f8\u5b9a\u671f\u91cd\u6d4b\u5206\u6790\u548c\u66f4\u65b0COA\uff0c\u4fdd\u8bc1\u4ea7\u54c1\u8d28\u91cf\u7684\u540c\u65f6\u4e5f\u4fdd\u8bc1\u5ba2\u6237\u7684\u6700\u957f\u6709\u6548\u671f\u3002<\/p>\n<p>\u6240\u6709\u4ea7\u54c1\u5305\u542b\u4e00\u4efd\u5168\u9762\u7684COA\u5206\u6790\u62a5\u544a\uff1a\u5168\u5149\u8c31\u5206\u6790\u3001\u50a8\u5b58\u6761\u4ef6\u3001\u4fdd\u8d28\u671f\u548c\u91cd\u6d4b\u5206\u6790\u65e5\u671f\u3001NMR\u548cHPLC-MS\u5206\u6790\u5316\u5b66\u7eaf\u5ea6\u3001\u540c\u4f4d\u7d20\u8d28\u91cf\u7eaf\u5ea6\uff0c\u6240\u6709\u6807\u51c6\u54c1\u53ef\u4ece1mg\u81f3100mg\u5206\u88c5\u5728\u8ba4\u8bc1\u7684\u7cbe\u786e\u79f0\u91cf\u7684\u50a8\u6837\u74f6\u4e2d\u3002<\/p>\n<p><img decoding=\"async\" class=\"alignnone size-full wp-image-463\" src=\"http:\/\/www.broadbio.com\/wp-content\/uploads\/2019\/12\/QQ\u622a\u56fe20191202103115.png\" alt=\"\" width=\"218\" height=\"81\" \/><\/p>\n<h2>5000+ \u7a33\u5b9a\u540c\u4f4d\u7d20\u6807\u8bb0\u4ea7\u54c1<br \/>\n\u63d0\u4f9b\u7a33\u5b9a\u540c\u4f4d\u7d20\u6807\u8bb0\u7684\u5b9a\u5236\u5408\u6210\u670d\u52a1\uff1a<\/h2>\n<p>&#8211; \u533b\u836f\u4e2d\u95f4\u4f53<br \/>\n&#8211; \u591a\u80bd<br \/>\n&#8211; \u751f\u7269\u6d3b\u6027<br \/>\n&#8211; \u7ba1\u63a7\u836f\u7269\u6807\u51c6\u54c1\uff08DEA\uff09<br \/>\n&#8211; \u4ee3\u8c22\u4ea7\u7269<br \/>\n&#8211; \u540c\u4f4d\u7d20\u6807\u8bb0\u53c2\u7167\u54c1<br \/>\n&#8211; \u519c\u836f<\/p>\n<p><span style=\"color: #ff0000;\"><strong>\u4ee5\u4e0b\u4e3aalsachim\u90e8\u5206\u4ea7\u54c1\u76ee\u5f55\uff0c\u66f4\u591a\u8be6\u7ec6\u4fe1\u606f\uff0c\u53ef\u4ee5\u6765\u7535\u54a8\u8be2\uff01<\/strong><\/span><\/p>\n<table width=\"1544\">\n<tbody>\n<tr>\n<td width=\"472\">[13C,2H3]-Tadalafil<\/td>\n<td width=\"173\">C2804<\/td>\n<td width=\"299\">1261364-86-6<\/td>\n<td width=\"600\">Cialis-13C-d3<\/td>\n<\/tr>\n<tr>\n<td>[2H3]-Estriol 3-sulfate 16-\u03b1-glucuronide<\/td>\n<td>C6315<\/td>\n<td>N\/A<\/td>\n<td>[2H3]-Estriol 3-sulfate 16-a-glucuronide<\/td>\n<\/tr>\n<tr>\n<td>[13C2,2H3,15N2]-Brotizolam<\/td>\n<td>C4099<\/td>\n<td>57801-81-7 unlabeled<\/td>\n<td>[13C6]-Lendormin<\/td>\n<\/tr>\n<tr>\n<td>[13C2,15N2]-Hexamethylenediamine dihydrochloride salt<\/td>\n<td>C7393<\/td>\n<td>6055-52-3 unlabeled<\/td>\n<td>[13C2, 15N2]-1,6-Hexanediamine dihydrochloride, [13C2, 15N2]-HMDA<\/td>\n<\/tr>\n<tr>\n<td>[13C6]-Licarbazepine<\/td>\n<td>C8231<\/td>\n<td>29331-92-8 unlabeled<\/td>\n<td>[13C6]-10,11-Dihydro-10-hydroxycarbamazepine<\/td>\n<\/tr>\n<tr>\n<td>[13C6]-6-Hydroxy Benzbromarone<\/td>\n<td>C7860<\/td>\n<td>152831-00-0 unlabeled<\/td>\n<td>[13C6]-Benzbromarone metabolite<\/td>\n<\/tr>\n<tr>\n<td>[2H5]-Selegiline oxalate salt<\/td>\n<td>C515<\/td>\n<td>2323-36-6 free base unlabeled<\/td>\n<td>[2H5]-R-(-)-Deprenyl hydrochloride<\/td>\n<\/tr>\n<tr>\n<td>[2H6]-DMST<\/td>\n<td>C7732<\/td>\n<td>66840-71-9 unlabeled<\/td>\n<td>[2H4]-4-Dimethylaminosulfotoluidide<\/td>\n<\/tr>\n<tr>\n<td>[2H8]-Terazosin Hydrochloride<\/td>\n<td>C7013<\/td>\n<td>1006718-20-2 free base<\/td>\n<td>[2H8]-1-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-4-[(tetrahydro-2-furanyl)carbonyl]piperazine hydrochloride, [2H8]-Abbott 45975<\/td>\n<\/tr>\n<tr>\n<td>[2H5]-N-Ethyloxamide<\/td>\n<td>C7398<\/td>\n<td>75235-35-7 unlabeled<\/td>\n<td>XP25547<\/td>\n<\/tr>\n<tr>\n<td>[13C,2H3]-Cediranib<\/td>\n<td>C4572<\/td>\n<td>288383-20-0 unlabeled<\/td>\n<td>Recentin, ZD 2171, AZD 2171<\/td>\n<\/tr>\n<tr>\n<td>[13C2,2H6]-Dabrafenib carboxylate dilithium salt<\/td>\n<td>C8275<\/td>\n<td>1195873-54-1 unlabeled free acid<\/td>\n<td><\/td>\n<\/tr>\n<tr>\n<td>[2H5]-Doripenem<\/td>\n<td>C8105<\/td>\n<td>364622-82-2 unlabeled<\/td>\n<td><\/td>\n<\/tr>\n<tr>\n<td>[13C,2H7]-Cangrelor<\/td>\n<td>C6563<\/td>\n<td>163706-06-7 unlabeled<\/td>\n<td><\/td>\n<\/tr>\n<tr>\n<td>[2H7]-Prothionamide<\/td>\n<td>C7344<\/td>\n<td>14222-60-7 unlabeled<\/td>\n<td><\/td>\n<\/tr>\n<tr>\n<td>[2H6]-Ceftazidime sodium salt<\/td>\n<td>C8506<\/td>\n<td>73547-61-2 unlabeled<\/td>\n<td><\/td>\n<\/tr>\n<tr>\n<td>[2H4]-Piroxicam<\/td>\n<td>C7032<\/td>\n<td>36322-90-4 unlabeled<\/td>\n<td><\/td>\n<\/tr>\n<tr>\n<td>[13C6]-Danshensu sodium salt<\/td>\n<td>C7974<\/td>\n<td>81075-52-7 unlabeled<\/td>\n<td><\/td>\n<\/tr>\n<tr>\n<td>[2H10]-Pitofenone hydrochloride salt<\/td>\n<td>C7029<\/td>\n<td>1248-42-6 unlabeled<\/td>\n<td><\/td>\n<\/tr>\n<tr>\n<td>[13C6]-4-Fluoro-2-(trifluoromethyl)aniline hydrochloride salt<\/td>\n<td>M993<\/td>\n<td>139291-82-0 unlabeled<\/td>\n<td><\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n","protected":false},"excerpt":{"rendered":"<p>\u6cd5\u56fdAlsaChim\u662f\u63d0\u4f9b\u9ad8\u54c1\u8d28\u7a33\u5b9a\u540c\u4f4d\u7d20\u5185\u6807\u548c\u4e34\u5e8a\u8d28\u8c31\u68c0\u6d4b\u8bd5\u5242\u76d2\u4ea7\u54c1\uff0c\u5176\u4e2d\u5305\u542b13C, 15N, 2H\u7684\u7a33\u5b9a [&hellip;]<\/p>\n","protected":false},"author":2,"featured_media":0,"comment_status":"closed","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"site-sidebar-layout":"default","site-content-layout":"","ast-site-content-layout":"","site-content-style":"default","site-sidebar-style":"default","ast-global-header-display":"","ast-banner-title-visibility":"","ast-main-header-display":"","ast-hfb-above-header-display":"","ast-hfb-below-header-display":"","ast-hfb-mobile-header-display":"","site-post-title":"","ast-breadcrumbs-content":"","ast-featured-img":"","footer-sml-layout":"","theme-transparent-header-meta":"","adv-header-id-meta":"","stick-header-meta":"","header-above-stick-meta":"","header-main-stick-meta":"","header-below-stick-meta":"","astra-migrate-meta-layouts":"default","ast-page-background-enabled":"default","ast-page-background-meta":{"desktop":{"background-color":"","background-image":"","background-repeat":"repeat","background-position":"center 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